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7-TM Receptors

A large proportion of commercially-available drugs target seven transmembrane (7-TM) receptors, of which a selection is offered by Carbosynth that are listed below. 7-TM receptors are the largest superfamily of cell surface receptors, also known as G-protein-coupled receptors (GPCRs). These receptors transduce signals from the extracellular space to the cytoplasm, via their transmembrane domains. Based on sequence homology, 7-TM receptors are classed into 6 groups: Class A (rhodopsin-like), Class B (secretin receptor family), Class C (metabotropic glutamate), Class D (fungal mating pheromone receptors), Class E (cyclic AMP receptors) and Class F (frizzled/smoothened).

Code Cas No Product Description
FA16904 447407-36-5

AC 42

Muscarinic (M1) receptor agonist BIO-X
BA17966 220556-69-4

ACEA

Cannabinoid (CB1) receptor agonist
BA166874 51037-30-0

Acipimox

Niacin receptor 1 (NIACR1) antagonist; lipid lowering BIO-R
FA31012 320345-99-1

Aclidinium bromide

Muscarinic antagonist; bronchodilator BIO-X
BA17967 229021-64-1

ACPA

CB1 cannabinoid receptor agonist
FA103122 851881-60-2

ADX 47273

Positive allosteric modulator of mGlu5 receptors BIO-X
BA166488 851881-59-9

(R)-ADX 47273

Positive allosteric modulator of metabotropic glutamate receptor mGluR5 BIO-X
BA167079 138112-76-2

Agomelatine

Melatonin agonist; 5-HT2B and 5-HT2C serotonin receptor antagonist BIO-X
BA164142 79561-22-1

Alarelin Acetate

Gonadotropin-releasing hormone agonist BIO-X
BA164143 18559-94-9

Albuterol

β2-adrenergic receptor agonist; bronchodilator BIO-R
FA17263 50293-90-8

(R)-Albuterol hydrochloride

β2-adrenergic receptor agonist; bronchodilator BIO-X
BA164388 51022-70-9

Albuterol sulfate

β-adrenergic receptor agonists BIO-X
BA164145 81403-80-7

Alfuzosin

α-adrenoceptor antagonist; treatment for benign prostatic hyperplasia BIO-X
FA150825 59338-87-3

Alizapride hydrochloride

Dopamine (D2) receptor antagonist BIO-X
BA166116 913358-93-7

Almorexant hydrochloride

Antagonist of orexin receptors OX1 and OX2 BIO-X
FA17315 154323-46-3

Almotriptan hydrochloride

Serotonin (5-HT) receptor agonist BIO-X
BA166465 122852-69-1

Alosetron hydrochloride

Serotonin 5-HT3 receptor antagonist BIO-X
FA31828 745-65-3

Alprostadil

Inhibits platelet aggregation; vasodilator BIO-X
BA164152 156053-89-3
170098-38-1

Alvimopan

Peripheral μ-opioid receptor antagonist; gastroprokinetic BIO-X
BA168613 251908-92-6

AM 1172

Inhibitor of anandamide uptake and FAAH
BA17338 183232-66-8

AM 251 NEW

CB1 cannabinoid receptor antagonist BIO-X
BA164153 177036-94-1

Ambrisentan

Endothelin A receptor antagonist; anti-hypertensive BIO-X
FA148913 155148-31-5

AMD 3100 octahydrochloride

Chemokine receptor CXCR4 antagonist BIO-X
FA104030 473719-41-4

AMG 487

CXCR3 antagonist BIO-X
BA164158 71675-85-9

Amisulpride

Dopamine D2/D3 receptor antagonist; anti-psychotic; BIO-X
BA164170 14028-44-5

Amoxapine

Serotonin (5-HT2) receptor antagonist; inhibits norepinephrine reuptake BIO-R
FA138836 2706-50-5

DL-Amphetamine hydrochloride

Analytic reference standard
FA162453 51-63-8

(+)-Amphetamine sulphate

Inhibits reuptake of catecholamines; stimulates central nervous system
FA17951 105219-56-5

Apafant

Platelet-activating factor antagonist BIO-X
BA165146 1268881-20-4

APD 371 NEW

Cannabinoid receptor CB2 agonist; analgesic BIO-X
BA166505 461443-59-4

Aplaviroc

Inhibits chemokine receptor CCR5; anti-viral activity against HIV BIO-X
BA164186 73218-79-8

Apraclonidine hydrochloride

α2-adrenoceptor agonist; anti-glaucoma agent BIO-X
BA164216 170729-80-3

Aprepitant

Antagonist of neurokinin-1 receptor; anti-emetic BIO-X
BA165448 733750-99-7

AR 231453

A potent and selective small molecule agonist of GPR119 BIO-X
BA171831 200815-49-2

Arformoterol tartrate

Bronchodilator
BA164218 129722-12-9

Aripiprazole

Partial agonist of dopamine (D2) and serotonin (5-HT1A) receptors BIO-X
BA45604 128007-31-8

Arvanil

CB1 cannabinoid receptor and vanilloid TRPV1 (VR1) agonist BIO-X
FA17998 65576-45-6

Asenapine

Inhibits dopamine, serotonin and adrenergic receptors BIO-X
BA167271 1282549-08-9

ASP 6432

Type 1 lysophosphatidic acid (LPA) receptor antagonist BIO-X
FA18002 68844-77-9

Astemizole

Histamine-1 receptor antagonist; hERG K+ channel blocker BIO-X
BA166036 29122-68-7

Atenolol

β-adrenoceptor blocker BIO-R
FA64946 104075-48-1

Atipamezole hydrochloride

α2-adrenoceptor antagonist BIO-X
FA40914 914453-95-5

Atosiban acetate

Oxytocin receptor antagonist BIO-X
FA29947 173937-91-2

Atrasentan

Endothelin receptor antagonist BIO-X
FA64949 195733-43-8

Atrasentan hydrochloride

Endothelin receptor antagonist BIO-X
FD102253 358970-97-5

AVE 1625

Antagonist of cannabinoid receptor CB1 BIO-X
FD41314 1204707-71-0

AZD 5069

CXCR2 antagonist BIO-X
BA164232 79307-93-0

Azelastine hydrochloride

Histamine-1 receptor antagonist; NFκB activator BIO-X
BA164233 147403-03-0

Azilsartan

Angiotensin II, type I receptor antagonist; anti-hypertensive BIO-X
FB18126 66514-99-6

(S)-Baclofen

GABA(B) agonist; anti-spastic agent; skeletal muscle relaxant
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